All Industries

Top Drug Discovery Companies

241 Drug Discovery companies, sorted by total funding raised.

CoSyne Therapeutics

Transforming drug discovery through polymathic AI

London, United Kingdom11–50Artificial Intelligence, Biotech
Seed·$8.8M·May 2022
SFA Therapeutics

Regulating the immune system to block cancer & autoimmune diseases

1–10Biotech, Drug Discovery
Bridge·$8.6M·Sep 2023
DreamFold AI

AI-powered protein discovery platform using generative ML to navigate protein space for novel med...

Montreal, CanadaArtificial Intelligence, Biotech
Series A·$8.5M·Mar 2025
Harmonic Discovery

Multi-targeted therapeutics to treat complex diseases

New York, United States1–10Biotech, Drug Discovery
Seed·$8.0M·Sep 2022
RxStrategiesAcquired

Comprehensive turnkey solution for Community Health Centers.

Boca Raton, United States11–50Drug Discovery, Healthcare
Venture Round·$7.8M·Jan 2003
Relevium Medical

Platform injectable gel based therapeutic for osteoarthritis

Galway, Ireland1–10Drug Discovery, Healthcare
Grant·$7.3M·Nov 2024
Known MedicineAcquired

Combining 3D cell culture & AI to translate drugs to clinical success

Salt Lake City, United States11–50Drug Discovery, Healthcare
Seed·$7.2M·Aug 2021
TenSixty Bio

Uses AI, cell models, and high-throughput assays to identify antibody targets and develop oncolog...

Cambridge, United States1–10Life Sciences, Artificial Intelligence
Series A·$7.2M·Aug 2022
Eigen Therapeutics

Develops ML-driven priming co-therapies and a discovery platform to improve targeted cancer treat...

Redwood City, United States1–10Biotech, Drug Discovery
Seed·$7.0M·Dec 2022
Lifepack

Indonesian digital pharmacy platform offering prescription and OTC medications, online doctor con...

Jakarta, Indonesia11–50Drug Discovery, Healthcare
Series A·$7.0M·Aug 2022
Bindwell

Building better pesticides with AI

San Francisco, United States1–10Agtech, Drug Discovery
Seed·$6.5M·Nov 2025
PB
Pepper Bio

Accelerates drug discovery for untreatable diseases

United StatesBiotech, Drug Discovery
Seed·$6.5M·Nov 2023
LEAH Labs

Living therapies for pets first, and their people next

Minneapolis, United States1–10Drug Discovery, Healthcare
Grant·$5.8M·Aug 2025
Sable Bio

AI-powered drug safety platform that generates toxicology insights from unstructured trial data t...

London, United Kingdom1–10Biotech, Drug Discovery
Seed·$5.7M·Feb 2026
Nanome

Virtual reality platform for collaborative molecular visualization and structure-based drug disco...

San Diego, United States11–50AR/VR, Biotech
Venture Round·$5.5M·Feb 2021
transcera

Venture-backed biotech translating Harvard lab discoveries into improved biologic drug delivery f...

Boston, United States1–10Biotech, Healthcare
Pre-seed·$5.4M·Jul 2021
Clock.Bio

Extending and improving the quality of life by reversing the harmful effects of time in our cells

Cambridge, United Kingdom1–10Biotech, Longevity
Seed·$5.3M·Oct 2024
Vincere Biosciences

Biotech developing small molecules targeting mitophagy to treat age-related diseases like Parkins...

United States1–10Biotech, Drug Discovery
Grant·$5.0M·Nov 2025
10x Science

AI platform for understanding complex molecules and prioritizing drug candidates.

San Francisco, United States1–10Artificial Intelligence, Drug Discovery
Seed·$4.8M·Apr 2026
Model Medicines

AI-driven drug discovery company using AI to model chemistry and human biology for medicine devel...

Artificial Intelligence, Biotech
Series A·$4.1M·Nov 2021
Zip Bio

Compressing biology to develop the next generation of therapies

Seattle, United States1–10Artificial Intelligence, Biotech
Seed·$4.0M·Sep 2024
Sequence Bio

Discovering the true signals of disease to power life-changing drugs.

St. John's, Canada51–200Drug Discovery, Genomics
Seed·$3.9M·Aug 2016
Menten AI

Menten AI designs peptide and protein therapeutics using quantum…

San Francisco, United States1–10Drug Discovery, Healthcare
Seed·$3.8M·Jun 2020
CellChorus

The dynamic single-cell analysis company

Houston, United States1–10Drug Discovery, Healthcare
Grant·$3.8M·Oct 2024
EPICYPHER, INC.

R&D company with 63 SBIR/STTR awards from Department of Health and Human Services.

DURHAM, United States51–200Biotech, Drug Discovery
Seed·$3.4M·Jun 2024