All Industries

Top Drug Discovery Companies

1,077 Drug Discovery companies, sorted by total funding raised.

Ankyra Therapeutics

Ankyra is developing cancer therapies based on localized cytokines that prime a systemic adaptive...

Boston, United States11–50Biotech, Drug Discovery
Series BTotal funding$45.0MNov 2021
Peptone

Biotechnology company designing small-molecule therapeutics that target intrinsically disordered ...

London, United Kingdom11–50Artificial Intelligence, Biotech
Series ATotal funding$42.5MJun 2022
MAPP BIOPHARMACEUTICAL, INC.

R&D company with 14 SBIR/STTR awards from Department of Health and Human Services, Department of ...

San Diego, United States51–200Biotech, Drug Discovery
GrantTotal funding$41.5MSep 2025
STAQ Pharma
Biotech, Drug Discovery
Series CTotal funding$41.0MMar 2022
Arpeggio Bio

Arpeggio Bio develops drugs targeting transcription factors using AI…

Boulder, United States11–50Biotech, Drug Discovery
Series BTotal funding$40.2MNov 2025
LUCA Science
Biotech, Drug Discovery
Series BTotal funding$40.1MJun 2022
Mantra Bio

Biotechnology company developing targeted exosome-based therapeutics using its proprietary REVEAL...

South San Francisco, United States11–50Biotech, Drug Discovery
Series ATotal funding$39.0MJan 2023
PBS Biotech
Biotech, Drug Discovery
Growth EquityTotal funding$39.0MJan 2025
Valinor Discovery

Frontier ML lab training virtual patient foundation models on multi-omic and clinical datasets to...

Salt Lake City, United States1–10Artificial Intelligence, Biotech
Venture RoundTotal funding$38.0MFeb 2026
AnagenexClosed

Drug discovery company combining DNA-encoded library technology with machine learning to identify...

South San Francisco, United StatesArtificial Intelligence, Biotech
Series ATotal funding$37.2MJun 2022
EPICYPHER, INC.

R&D company with 63 SBIR/STTR awards from Department of Health and Human Services.

Durham, United States51–200Biotech, Deep Tech
GrantTotal funding$36.8MAug 2025
Shiru

Shiru harnesses the power of AI, bioinformatics, and precision biology to revolutionize ingredien...

Emeryville, United States1–10Agtech, Artificial Intelligence
Series BTotal funding$36.6MNov 2024
Beekeeper's Naturals

Bee propolis-powered wellness and supplement brand offering clean, natural immunity and energy pr...

Canada11–50Healthcare, Drug Discovery
Series DTotal funding$36.2MMar 2024
Permanence Bio

Developing therapeutics to stop mutations to prevent cancer

San Francisco, United States1–10Biotech, Drug Discovery
Series ATotal funding$35.0MJan 2026
Draupnir Bio

Draupnir Bio is a Danish biotechnology company developing small molecule therapeutics to transfor...

Biotech, Drug Discovery
Series ATotal funding$35.0M
InspheroAcquired

modernizing drug discovery

Schlieren, Switzerland51–200Biotech, Drug Discovery
Venture RoundTotal funding$35.0MMar 2023
Transcripta Bio

AI-powered drug discovery for neurological diseases

Palo Alto, United StatesArtificial Intelligence, Biotech
Series ATotal funding$34.0MJul 2026
C4U CORPORATION

Medical (medical devices, drug discovery) - Middle to Growth

Osaka, JapanBiotech, Drug Discovery
GrantTotal funding$33.5MJun 2025
FLUGEN INC

R&D company with 4 SBIR/STTR awards from Department of Health and Human Services.

Madison, United States11–50Biotech, Healthcare
GrantTotal funding$33.2MJul 2021
Transcode Therapeutics, Inc.

R&D company with 3 SBIR/STTR awards from Department of Health and Human Services.

Boston, United States1–10Biotech, Drug Discovery
Series BTotal funding$33.0MOct 2025
Aspen RxHealth

Technology platform connecting health plans, providers, and life science companies with an on-dem...

Tampa, United StatesDigital Health, Drug Discovery
Series BTotal funding$32.0MJan 2021
Javelin PharmaceuticalsAcquired
Biotech, Developer Tools
Corporate RoundTotal funding$32.0MNov 2005
Reverie LabsClosed

Engineering next-generation, brain-penetrant cancer therapies.

Cambridge, United States11–50Biotech, Drug Discovery
SeedTotal funding$32.0M
Envisagenics

AI-driven biotechnology company discovering RNA splicing targets and developing therapeutics for ...

Long Island City, United States11–50Artificial Intelligence, Biotech
Series BTotal funding$31.4MJun 2024
Sorriso Pharmaceuticals

Sorriso Pharmaceuticals is a biotechnology company advancing a pipeline of disease-modifying anti...

Sandy, United States1–10Biotech, Drug Discovery
Series ATotal funding$31.0MDec 2021