Iterion Therapeutics
- Website
- iteriontherapeutics.com
- Total Funding
- $24.1M
- Last Round
- $7.1M GrantNov 2025
- Rounds
- 2
About
Iterion Therapeutics is developing tegavivint, a novel small-molecule inhibitor that binds to TBL1 and disrupts the interaction between beta-catenin and TBL1, promoting degradation of nuclear beta-catenin and preventing transcription of Wnt/beta-catenin targeted oncogenes. Preclinical studies have shown tegavivint inhibits beta-catenin activity without overt toxicity and is not affected by CTNNB1 gain-of-function mutations typically found in cancer cells. In parallel with the tegavivint program, Iterion has ongoing R&D programs investigating and developing second-generation TBL1 inhibitors.
Summary
Iterion Therapeutics is a Biotech company. It has raised $24.1M in total across 2 rounds, most recently a $7.1M Grant round in Nov 2025. Investors include Cancer Prevention and Research Institute of Texas, Sante Ventures and Lumira Ventures.
Funding History
Nov 2025
Sign up to see all 2 rounds
Series B through Grant — per-round amounts, valuations, and who invested in each round.
Investors
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